Drug class

Antineoplas-Tissue Factor Directed Ab-Microtub Disrupt Conj

The phrase "Antineoplas-Tissue Factor Directed Ab-Microtub Disrupt Conj" is an abbreviated formulary or administrative classification describing antineoplastic tissue factor-directed antibody and microtubule disruptor conjugates. Read more about Antineoplas-Tissue Factor Directed Ab-Microtub Disrupt Conj

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About Antineoplas-Tissue Factor Directed Ab-Microtub Disrupt Conj.

The phrase "Antineoplas-Tissue Factor Directed Ab-Microtub Disrupt Conj" is an abbreviated formulary or administrative classification describing antineoplastic tissue factor-directed antibody and microtubule disruptor conjugates.

Rather than a broad pharmacological family, this specialized category currently represents targeted antibody-drug conjugates exemplified by tisotumab vedotin.

Agents in this class consist of a monoclonal antibody targeting cell-surface tissue factor linked to an antimitotic cytotoxic payload, such as monomethyl auristatin E, which inhibits tubulin polymerization and causes cell cycle arrest and apoptosis upon cellular internalization.

Therapeutics in this group are primarily utilized in oncology for the treatment of adult patients with recurrent or metastatic cervical cancer that has progressed on or following systemic chemotherapy.